Channeling teamwork: ATP and lipids cooperate to gate P2X receptors

P2X receptor structures resolved in a lipid environment reveal how subtype-specific ligand recognition, drug sensitivity, and channel gating are coupled.

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Publication Details

Journal
Science Advances
Published
2026-05-27
DOI
https://doi.org/10.1126/sciadv.aei2053
Primary Topic
Adenosine and Purinergic Signaling
Type
article
Field-Weighted Citation Impact
0.00
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article

Channeling teamwork: ATP and lipids cooperate to gate P2X receptors

Frank Bosmans, Toshimitsu Kawate
Science Advances
Adenosine and Purinergic Signaling
article

Channeling teamwork: ATP and lipids cooperate to gate P2X receptors

Frank Bosmans, Toshimitsu Kawate
article en

Abstract

P2X receptor structures resolved in a lipid environment reveal how subtype-specific ligand recognition, drug sensitivity, and channel gating are coupled.

Science AdvancesVol. 12(22)
Vrije Universiteit Brussel (BE), Cornell University (US), Ghent University (BE)
Openalex Percentile: Top 8%
Adenosine and Purinergic Signaling
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