Hypervalent Iodine(III)-Mediated Oxidative C–H Amination of Phenols and Anilines with Azoles
COOH as the terminal oxidant-acid pair delivers comparable efficiency. This operationally simple protocol complements palladium- or copper-catalyzed methods by eliminating aryl-halide preactivation and transition metals.
Authors
- Koji Morimoto (ORCID: https://orcid.org/0000-0001-5019-5158)
- Yasuyuki Kita (ORCID: https://orcid.org/0000-0002-2482-0551)
- Kana Yanase
- Toshifumi Dohi (ORCID: https://orcid.org/0000-0002-2812-9581)
Institutions
- Ritsumeikan University (JP)
Publication Details
- Journal
- Organic Letters
- Published
- 2026-04-22
- DOI
- https://doi.org/10.1021/acs.orglett.6c01148
- Primary Topic
- Catalytic C–H Functionalization Methods
- Type
- article
- Field-Weighted Citation Impact
- 0.00
Funders
- Ministry of Education, Culture, Sports, Science and Technology
- Japan Society for the Promotion of Science