Novel Dihydroisoquinolinone-Amide Compounds as GIPR Agonists for Treating Type 2 Diabetes Mellitus and Obesity

Provided herein are novel dihydroisoquinolinone-amide compounds as GIPR agonists, pharmaceutical compositions, use of such compounds in treating type 2 diabetes mellitus and obesity, and processes for preparing such compounds.

Authors

Publication Details

Journal
ACS Medicinal Chemistry Letters
Published
2026-04-16
DOI
https://doi.org/10.1021/acsmedchemlett.6c00175
Primary Topic
Pharmacology and Obesity Treatment
Type
article
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article

Novel Dihydroisoquinolinone-Amide Compounds as GIPR Agonists for Treating Type 2 Diabetes Mellitus and Obesity

Ram W. Sabnis
ACS Medicinal Chemistry Letters
Pharmacology and Obesity Treatment
article

Novel Dihydroisoquinolinone-Amide Compounds as GIPR Agonists for Treating Type 2 Diabetes Mellitus and Obesity

Ram W. Sabnis
article en

Abstract

Provided herein are novel dihydroisoquinolinone-amide compounds as GIPR agonists, pharmaceutical compositions, use of such compounds in treating type 2 diabetes mellitus and obesity, and processes for preparing such compounds.

ACS Medicinal Chemistry Letters
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Pharmacology and Obesity Treatment
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Novel Dihydroisoquinolinone-Amide Compounds as GIPR Agonists for Treating Type 2 Diabetes Mellitus and Obesity — Ram W. Sabnis · ACS Medicinal Chemistry Letters (2026) | TGRS Research Map | TGRS