Trifluoromethylthio and Trifluoromethyl Functionalization of Endomorphin-1 Enhances its Hydrophobicity and Plasma Stability while Preserving its Affinity for the μ-Opioid Receptor
Authors
Steven Ballet (ORCID: https://orcid.org/0000-0003-4123-1641)
Brian J. Holleran (ORCID: https://orcid.org/0000-0003-3136-1928)
Faculty of Medicine and Health, University of Sydney
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article
Trifluoromethylthio and Trifluoromethyl Functionalization of Endomorphin-1 Enhances its Hydrophobicity and Plasma Stability while Preserving its Affinity for the μ-Opioid Receptor
Steven Ballet, Brian J. Holleran, Jure Gregorc, Grégory Chaume et al.
Journal
The Journal of Organic Chemistry
Topics
Neuropeptides and Animal Physiology
article
Trifluoromethylthio and Trifluoromethyl Functionalization of Endomorphin-1 Enhances its Hydrophobicity and Plasma Stability while Preserving its Affinity for the μ-Opioid Receptor
Steven Ballet, Brian J. Holleran, Jure Gregorc, Grégory Chaume, Karine Guitot, Louis Gendron, Jernej Iskra, Thierry Brigaud, Jolien De Neve, Nathalie Lensen
article en
Abstract
No abstract available for this paper.
Publication Tag
The Journal of Organic ChemistryVol. 91(16)
Institutions
Centre National de la Recherche Scientifique (FR), Vrije Universiteit Brussel (BE), Université de Sherbrooke (CA), University of Ljubljana (SI), Université Paris-Saclay (FR), CY Cergy Paris Université (FR), Bioengineering Center (RU)
Funders
Université de Sherbrooke, Agence Nationale de la Recherche, Fonds Wetenschappelijk Onderzoek, Javna Agencija za Raziskovalno Dejavnost RS, Vrije Universiteit Brussel, Centre National de la Recherche Scientifique, Université Paris-Saclay, Univerza v Ljubljani, Vlaamse regering, Faculty of Medicine and Health, University of Sydney