Micron-Scale 2D Antibody Arrays for HER2 Signaling Blockade and Cancer Therapy

Monoclonal antibodies (mAbs) targeting the human epidermal growth factor receptor 2 (HER2) are widely used in the treatment of breast, gastric, and other solid tumors. However, rapid HER2 endocytosis and recycling contribute to low response rates and treatment resistance. Here, we introduce RhuA-P, a self-assembling protein that forms uniform, micron-sized 2D arrays (2.4 × 2.4 μm) featuring spatially addressable Protein G sites for mAb conjugation. This design allows control over antibody density (22-274 molecules per array) and intermolecular spacing (57-230 nm). We show that trastuzumab (TmAb) arrays templated on RhuA-P inhibit HER2 dimerization, cluster HER2 into micron-scale inactive domains dictated by the 2D TmAb geometry, and prolong receptor membrane retention by blocking endocytosis. This sustained blockade of HER2 signaling induces oxidative stress and triggers potent apoptosis. In a murine breast cancer model, TmAb arrays exhibited superior antitumor efficacy compared to free TmAb. Moreover, the modular design of RhuA-P makes it a versatile platform for assembling other clinically relevant mAbs─such as anti-PD-1 and anti-PD-L1 antibodies─offering a generalized strategy for enhancing antibody-based therapies.

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Publication Details

Journal
Journal of the American Chemical Society
Published
2026-02-23
DOI
https://doi.org/10.1021/jacs.5c22627
Primary Topic
Monoclonal and Polyclonal Antibodies Research
Type
article
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article

Micron-Scale 2D Antibody Arrays for HER2 Signaling Blockade and Cancer Therapy

Xiangyu Wu, Sisi Ling, Qian Chen, Tingfeng Yao et al.
Journal of the American Chemical Society
Monoclonal and Polyclonal Antibodies Research
article

Micron-Scale 2D Antibody Arrays for HER2 Signaling Blockade and Cancer Therapy

Xiangyu Wu, Sisi Ling, Qian Chen, Tingfeng Yao, Yong Li, Mingming Du, Xiang Zhong, G. Chen, Qiangbin Wang, Yuefei Wang, Jiang Jiang
article en

Abstract

Monoclonal antibodies (mAbs) targeting the human epidermal growth factor receptor 2 (HER2) are widely used in the treatment of breast, gastric, and other solid tumors. However, rapid HER2 endocytosis and recycling contribute to low response rates and treatment resistance. Here, we introduce RhuA-P, a self-assembling protein that forms uniform, micron-sized 2D arrays (2.4 × 2.4 μm) featuring spatially addressable Protein G sites for mAb conjugation. This design allows control over antibody density (22-274 molecules per array) and intermolecular spacing (57-230 nm). We show that trastuzumab (TmAb) arrays templated on RhuA-P inhibit HER2 dimerization, cluster HER2 into micron-scale inactive domains dictated by the 2D TmAb geometry, and prolong receptor membrane retention by blocking endocytosis. This sustained blockade of HER2 signaling induces oxidative stress and triggers potent apoptosis. In a murine breast cancer model, TmAb arrays exhibited superior antitumor efficacy compared to free TmAb. Moreover, the modular design of RhuA-P makes it a versatile platform for assembling other clinically relevant mAbs─such as anti-PD-1 and anti-PD-L1 antibodies─offering a generalized strategy for enhancing antibody-based therapies.

Journal of the American Chemical SocietyVol. 148(9)
University of Science and Technology of China (CN), Chinese Academy of Sciences (CN), ShanghaiTech University (CN), Suzhou Institute of Nano-tech and Nano-bionics (CN), University of Chinese Academy of Sciences (CN)
Good health and well-being
Openalex Percentile: Top 47%
Monoclonal and Polyclonal Antibodies Research
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