Novel Compounds as ARNT Degraders for Treating Cancer, in Particular, Hematological Cancer

Provided herein are novel compounds as ARNT degraders, pharmaceutical compositions, use of such compounds in treating cancer, in particular, hematological cancer, and processes for preparing such compounds.

Authors

Publication Details

Journal
ACS Medicinal Chemistry Letters
Published
2026-01-05
DOI
https://doi.org/10.1021/acsmedchemlett.5c00777
Primary Topic
Electron Spin Resonance Studies
Type
article
Field-Weighted Citation Impact
0.00
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article

Novel Compounds as ARNT Degraders for Treating Cancer, in Particular, Hematological Cancer

Ram W. Sabnis
ACS Medicinal Chemistry Letters
Electron Spin Resonance Studies
article

Novel Compounds as ARNT Degraders for Treating Cancer, in Particular, Hematological Cancer

Ram W. Sabnis
article en

Abstract

Provided herein are novel compounds as ARNT degraders, pharmaceutical compositions, use of such compounds in treating cancer, in particular, hematological cancer, and processes for preparing such compounds.

ACS Medicinal Chemistry LettersVol. 17(2)
Openalex Percentile: Top 98%
Electron Spin Resonance Studies
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Novel Compounds as ARNT Degraders for Treating Cancer, in Particular, Hematological Cancer — Ram W. Sabnis · ACS Medicinal Chemistry Letters (2026) | TGRS Research Map | TGRS