Copper-Catalyzed Diamination of Alkenes using <i>o</i>‑Benzoylhydroxylamines to Access the Four Azaindoline\nFamilies

A mild\nand efficient method for the copper-catalyzed diamination\nof alkenes is described. In this reaction, <i>o</i>-benzoylhydroxylamine\nserves as an electrophilic nitrogen source for the regioselective\nformation of C–N bonds. This transformation provides a novel\nstrategy for synthesizing all four isomeric 2,3-disubstituted azaindoline\nfamilies and offers a wide substrate scope.

Publication Details

Journal
Figshare
Published
2024-10-04
DOI
https://doi.org/10.1021/acs.orglett.4c02585.s001
Primary Topic
Catalytic C–H Functionalization Methods
Type
article
Field-Weighted Citation Impact
0.00
Controls
|||
ALL TIME
JAN
FEB
MAR
APR
MAY
JUN
JUL
AUG
SEP
OCT
article

Copper-Catalyzed Diamination of Alkenes using o‑Benzoylhydroxylamines to Access the Four Azaindoline\nFamilies

Figshare
Catalytic C–H Functionalization Methods
article

Copper-Catalyzed Diamination of Alkenes using o‑Benzoylhydroxylamines to Access the Four Azaindoline\nFamilies

article en

Abstract

A mild\nand efficient method for the copper-catalyzed diamination\nof alkenes is described. In this reaction, <i>o</i>-benzoylhydroxylamine\nserves as an electrophilic nitrogen source for the regioselective\nformation of C–N bonds. This transformation provides a novel\nstrategy for synthesizing all four isomeric 2,3-disubstituted azaindoline\nfamilies and offers a wide substrate scope.

Figshare
Openalex Percentile: Top 60%
Catalytic C–H Functionalization Methods
DOIOpen Access PDFOpenAlex
AI Navigator

Ask Laika to Summarize, Analyze, and Connect papers live on the map.

Summarize Papers & Methodologies

Extract key findings, datasets, and comparative methods across publications.

Benchmark Rankings & Visual Analytics

Rank top research institutions, authors, funders, topics, and journals by Field-Weighted Citation Impact (FWCI) and paper volume with instant charts.

Connect Distant Disciplines

Bridge topological clusters on the map to find hidden collaborative intersections.

Copper-Catalyzed Diamination of Alkenes using <i>o</i>‑Benzoylhydroxylamines to Access the Four Azaindoline\nFamilies · Figshare (2024) | TGRS Research Map | TGRS