Monitoring the plasma concentration of ripretinib and its metabolites in Chinese patients with gastrointestinal stromal tumors in a real‐life setting

Ripretinib and its metabolites maintained consistent plasma concentrations in Chinese patients with advanced GIST. Furthermore, a trough ripretinib concentration >475 ng/mL was associated with extended survival.

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Publication Details

Journal
Cancer
Published
2025-12-01
DOI
https://doi.org/10.1002/cncr.70149
Primary Topic
Gastrointestinal Tumor Research and Treatment
Type
article
Field-Weighted Citation Impact
0.00

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article

Monitoring the plasma concentration of ripretinib and its metabolites in Chinese patients with gastrointestinal stromal tumors in a real‐life setting

Ye Zhou, Hao Xu, Zekuan Xu, Qiang Zhang et al.
Cancer
Gastrointestinal Tumor Research and Treatment
article

Monitoring the plasma concentration of ripretinib and its metabolites in Chinese patients with gastrointestinal stromal tumors in a real‐life setting

Ye Zhou, Hao Xu, Zekuan Xu, Qiang Zhang, Rui Wang, Ming Wang, Yongqing Wang, Fengyuan Li, Xin Wu, Yongjian Zhou, Xiaofeng Sun, Haoran Qian, Linsen Zhou, Luning Sun
article en

Abstract

Ripretinib and its metabolites maintained consistent plasma concentrations in Chinese patients with advanced GIST. Furthermore, a trough ripretinib concentration >475 ng/mL was associated with extended survival.

CancerVol. 131(S3)
Fujian Medical University (CN), Shanghai Medical College of Fudan University (CN), Shanghai Jiao Tong University (CN), Nantong University (CN), Renji Hospital (CN), Sir Run Run Shaw Hospital (CN), Chinese PLA General Hospital (CN), Fudan University Shanghai Cancer Center (CN), Nanjing Drum Tower Hospital (CN), Ministry of Education (KR), Yancheng First People's Hospital (CN), Yancheng Third People's Hospital (CN), Jiangsu Cancer Hospital (CN), Yancheng Second People's Hospital (CN), Jiangsu Province Hospital (CN), Union Hospital (CN), Zhejiang University (CN), Nanjing Medical University (CN)
National Natural Science Foundation of China, Government of Jiangsu Province, Natural Science Foundation of Jiangsu Province, Nanjing Medical University, Chinese Society of Clinical Oncology, Priority Academic Program Development of Jiangsu Higher Education Institutions
Openalex Percentile: Top 45%
Gastrointestinal Tumor Research and Treatment
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