In vitro and in silico evaluation of synthetic compounds derived from bi-triazoles against asexual and sexual forms of Plasmodium falciparum
Overall, the in vitro and in silico results showed that bi-triazole compounds may guide new biological investigation for malaria, enabling the identification and development of more active and selective antimalarial agents.
Authors
- Sabrina Baptista Ferreira (ORCID: https://orcid.org/0000-0002-5363-0888)
- Aurileya de Jesus Gouveia (ORCID: https://orcid.org/0000-0001-6360-3026)
- Jansen Fernandes Medeiros (ORCID: https://orcid.org/0000-0003-4196-8985)
- Ana Paula de Azevedo dos Santos (ORCID: https://orcid.org/0000-0003-4005-6263)
- Carlos R. Kaiser (ORCID: https://orcid.org/0000-0002-2132-1351)
- Carolina Bioni Garcia Teles (ORCID: https://orcid.org/0000-0002-4529-2137)
- Norton Rubens Diunior Lucas Pejara Rossi (ORCID: https://orcid.org/0000-0003-1980-575X)
- Welington da Silva Paula do Nascimento (ORCID: https://orcid.org/0000-0001-6935-952X)
- Marcinete Latorre Almeida (ORCID: https://orcid.org/0000-0002-8963-5939)
- Saara Neri Fialho
- Quelli Larissa Oliveira de Santana (ORCID: https://orcid.org/0000-0002-8940-4022)
- Amália dos Santos Ferreira
- Minelly Azevedo da Silva (ORCID: https://orcid.org/0000-0002-6052-6341)
- Leandro do Nascimento Martinez (ORCID: https://orcid.org/0000-0003-0887-4784)
- Maísa da Silva Araújo (ORCID: https://orcid.org/0000-0003-3607-0433)
- Nuna Araújo
Institutions
- Universidade Federal do Rio de Janeiro (BR)
- Universidade Federal de Rondônia (BR)
- Instituto Federal de Educação, Ciência e Tecnologia de Rondônia (BR)
- Centro Universitário São Lucas (BR)
- Fundação Oswaldo Cruz (BR)
Publication Details
- Journal
- Malaria Journal
- Published
- 2025-03-04
- DOI
- https://doi.org/10.1186/s12936-025-05297-7
- Primary Topic
- Click Chemistry and Applications
- Type
- article
- Field-Weighted Citation Impact
- 0.00
Funders
- Bill and Melinda Gates Foundation
- Coordenação de Aperfeiçoamento de Pessoal de Nível Superior
- Conselho Nacional de Desenvolvimento Científico e Tecnológico
- Ministério da Saúde
- Fundação Oswaldo Cruz