Biological Evaluation and Computational Modelling Studies on N-acyl Hydrazone and 2,5-Disubstituted 1,3,4-Oxadiazole Derivatives as Non-toxic Antimicrobial Agents
Further exploration of molecular determinants revealed favourable drug-like properties, highlighting the potential of these molecules for subsequent hit-to-lead optimization studies.
Authors
- Semra Şardaş (ORCID: https://orcid.org/0000-0001-5456-8636)
- Hatice Başpınar Küçük (ORCID: https://orcid.org/0000-0002-1735-6260)
- Mattia Mori (ORCID: https://orcid.org/0000-0003-2398-1254)
- Ayşe Şeyma Büyük (ORCID: https://orcid.org/0000-0001-8934-0359)
- Martina Fiabane (ORCID: https://orcid.org/0009-0009-2438-9018)
- Nil Kaya (ORCID: https://orcid.org/0000-0002-1444-4935)
- Betül Giray
Institutions
- University of Siena (IT)
- Istanbul University-Cerrahpaşa (TR)
- Istinye University (TR)
- Istanbul University (TR)
Publication Details
- Journal
- Current Pharmaceutical Design
- Published
- 2025-02-12
- DOI
- https://doi.org/10.2174/0113816128361524250131110036
- Citations
- 3
- Primary Topic
- Synthesis and biological activity
- Type
- article
- Field-Weighted Citation Impact
- 2.81