QSAR Studies on a Class of Benzofuranene Cyanide Derivatives as Potential Inhibitors Targeting Staphylococcus aureus Sortase A
In this study, two quantitative structure-activity relationship models were successfully established to predict the inhibitory activity of a series of compounds targeting Staphylococcus aureus Sortase A, providing insights for further development of novel anti-Staphylococcus aureus drugs.
Authors
- Jinqiu Zhang (ORCID: https://orcid.org/0000-0002-5192-2182)
- Shaodong Fu (ORCID: https://orcid.org/0009-0008-0330-4399)
- Yawei Qiu (ORCID: https://orcid.org/0009-0007-4306-4767)
- Jinfeng Miao (ORCID: https://orcid.org/0000-0001-6229-3767)
- Bo Yang (ORCID: https://orcid.org/0000-0002-6156-8957)
Institutions
- Nanjing Agricultural University (CN)
- Jiangsu Academy of Agricultural Sciences (CN)
Publication Details
- Journal
- Current Medicinal Chemistry
- Published
- 2024-09-03
- DOI
- https://doi.org/10.2174/0109298673300334240821041349
- Primary Topic
- Biochemical and Structural Characterization
- Type
- article
- Field-Weighted Citation Impact
- 0.00